Chemical Structure : GB83
CAS No.:
1252806-86-2
GB83
(PAR2 antagonist GB83)
Catalog No. : PC-61618Not For Human Use, Lab Use Only.
GB83 is a selective, reversible PAR2 (Protease-activated receptor 2) antagonist with IC50 of 2 uM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6161801
Biological Activity
GB83 is a selective, reversible PAR2 (Protease-activated receptor 2) antagonist with IC50 of 2 uM.
Physicochemical Properties
M.Wt
548.72
Formula
C32H44N4O4
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
N-((S)-3-cyclohexyl-1-((2S,3S)-1-(2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl)-3-methyl-1-oxopentan-2-ylamino)-1-oxopropan-2-yl)isoxazole-5-carboxamide
References
1. Barry GD, et al. J Med Chem.
2. Bukowska A, et al. Eur J Pharmacol.
3. Muley MM, et al. Br J Pharmacol.
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