GCN2 activator-1

Chemical Structure : GCN2 activator-1

Catalog No.: PC-28682Not For Human Use, Lab Use Only.

GCN2 activator-1 (Compound 20) is a GCN1-independent small molecule GCN2 activator, binds within the ATP-pocket of GCN2, inhibits PKR (EIF2AK2) in vitro with IC50 of 3.75 uM.

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Biological Activity

GCN2 activator-1 (Compound 20) is a GCN1-independent small molecule GCN2 activator, binds within the ATP-pocket of GCN2, inhibits PKR (EIF2AK2) in vitro with IC50 of 3.75 uM.

Physicochemical Properties

M.Wt	290.36
Formula	C11H10N6S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4'-Methyl-N2-(pyrimidin-2-yl)-[4,5'-bithiazole]-2,2'-diamine

References

1. JiaYi Zhu, et al. Elife. 2026 Oct 27:14:RP108590.

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GCN2 activator-1

Biological Activity

Physicochemical Properties

References

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