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Chemical Structure : GNE-886
Catalog No.: PC-62550Not For Human Use, Lab Use Only.
GNE-886 is a potent and selective CECR2 bromodomain inhibitor with IC50 of 16 nM.
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GNE-886 is a potent and selective CECR2 bromodomain inhibitor with IC50 of 16 nM.
GNE-886 shows a wide selectivity over the 40 bromodomains, >100-fold selectivity over BRD9, BRD7, TAF1(2), and BRD4(1).
GNE-886 has a highly favorable measured kinetic solubility of 122 uM and is an appropriate in vitro tool compound for the CECR2 bromodomain.
| M.Wt | 498.587 | |
| Formula | C28H30N6O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Crawford TD, et al. ACS Med Chem Lett. 2017 Jun 1;8(7):737-741.
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