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GPR54 antagonist 9l

Chemical Structure : GPR54 antagonist 9l

CAS No.: 925932-64-5

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GPR54 antagonist 9l

Catalog No.: PC-21176Not For Human Use, Lab Use Only.

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.
GPR54 antagonist 9l exhibits fully potent antagonist activity (IC50=0.46 μM) in cellular Ca2+ mobilization assays.

Physicochemical Properties

M.Wt 521.93
Formula C26H21ClFN5O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-{4-[3-(beta-Alanylamino)phenyl]-3-cyano-6-(4-fluoro-2-hydroxyphenyl)pyridin-2-yl}furan-2-carboxamide hydrochloride

References

1. Kobayashi T, et al. Bioorg Med Chem. 2010 Jun 1;18(11):3841-59.

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