GPR54 antagonist 9l

Chemical Structure : GPR54 antagonist 9l

Catalog No.: PC-21176Not For Human Use, Lab Use Only.

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.

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Biological Activity

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.
GPR54 antagonist 9l exhibits fully potent antagonist activity (IC50=0.46 μM) in cellular Ca2+ mobilization assays.

Physicochemical Properties

M.Wt	521.93
Formula	C26H21ClFN5O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-{4-[3-(beta-Alanylamino)phenyl]-3-cyano-6-(4-fluoro-2-hydroxyphenyl)pyridin-2-yl}furan-2-carboxamide hydrochloride

References

1. Kobayashi T, et al. Bioorg Med Chem. 2010 Jun 1;18(11):3841-59.

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