Chemical Structure : GPR54 antagonist 9l
Catalog No.: PC-21176Not For Human Use, Lab Use Only.
GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.
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GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.
GPR54 antagonist 9l exhibits fully potent antagonist activity (IC50=0.46 μM) in cellular Ca2+ mobilization assays.
M.Wt | 521.93 | |
Formula | C26H21ClFN5O4 | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Kobayashi T, et al. Bioorg Med Chem. 2010 Jun 1;18(11):3841-59.
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