You are here:Home-Chemical Inhibitors & Agonists-Others-Other Targets-GPR54 antagonist 9l
GPR54 antagonist 9l

Chemical Structure : GPR54 antagonist 9l

CAS No.: 925932-64-5

GPR54 antagonist 9l

Catalog No.: PC-21176Not For Human Use, Lab Use Only.

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.

Packing Price Stock Quantity
50 mg Get quote
100 mg Get quote
200 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GPR54 antagonist 9l is a potent, selective, small molecule antagonist of GPR54 with IC50 of 3.7 nM (human GPR54) in receptor binding assays.
GPR54 antagonist 9l exhibits fully potent antagonist activity (IC50=0.46 μM) in cellular Ca2+ mobilization assays.

Physicochemical Properties

M.Wt 521.93
Formula C26H21ClFN5O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-{4-[3-(beta-Alanylamino)phenyl]-3-cyano-6-(4-fluoro-2-hydroxyphenyl)pyridin-2-yl}furan-2-carboxamide hydrochloride

References

1. Kobayashi T, et al. Bioorg Med Chem. 2010 Jun 1;18(11):3841-59.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: