GPR56 agonist 36

Chemical Structure : GPR56 agonist 36

Catalog No.: PC-20909Not For Human Use, Lab Use Only.

GPR56 agonist 36 is a potent selective agonist of adhesion GPCR ADGRG1/GPR56 with EC50 of 2.95 uM.

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Biological Activity

GPR56 agonist 36 is a potent selective agonist of adhesion GPCR ADGRG1/GPR56 with EC50 of 2.95 uM.
GPR56 agonist 36 activates GPR56 F385A/M389A and GPR56 L388A/M389A double TA mutant holoreceptors.
GPR56 agonist 36 shows exclusive specificity for GPR56 in a small panel of adhesion GPCRs and two class A GPCRs. ADGRG5/GPR114, ADGRG3/GPR97, and ADGRG1/GPR56 are from the same adhesion GPCR subfamily.

Physicochemical Properties

M.Wt	432.36
Formula	C22H26BrNO3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C(C1=C(C)NC2=C(C(CC(C)(C)C2)=O)C1C3=CC=CC=C3Br)OC(C)C

References

1. Alexander L Vizurraga, et al. Mol Pharmacol. 2023 Jun 8;MOLPHARM-AR-2023-000688.

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GPR56 agonist 36

Biological Activity

Physicochemical Properties

References

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