GPR61 inverse agonist 15

Chemical Structure : GPR61 inverse agonist 15

Catalog No.: PC-26403Not For Human Use, Lab Use Only.

GPR61 inverse agonist 15 is a potent, selective, and brain-penetrant GPR61 inverse agonist with cAMP functional IC50 of 6.2 nM and 20 nM for human and mouse GPR61 respectively.

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Biological Activity

GPR61 inverse agonist 15 is a potent, selective, and brain-penetrant GPR61 inverse agonist with cAMP functional IC50 of 6.2 nM and 20 nM for human and mouse GPR61 respectively.

Physicochemical Properties

M.Wt	454.88
Formula	C18H17ClF2N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(5-Chloro-4,6-dimethylpyrimidin-2-yl)-6-(((3,5-difluoropyridin-4-yl)methyl)amino)-2-methylpyridine-3-sulfonamide

References

1. Fisher EL, et al. J Med Chem. 2026 Mar 15. doi: 10.1021/acs.jmedchem.6c00081.

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