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GPR7 antagonist 21a

Chemical Structure : GPR7 antagonist 21a

CAS No.: 2648124-49-4

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GPR7 antagonist 21a

Catalog No.: PC-38613Not For Human Use, Lab Use Only.

GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

    Physicochemical Properties

    M.Wt 397.182
    Formula C17H9Cl2F3N4
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    2-(2,6-dichloro-4-(1H-pyrazol-4-yl)phenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazole

    References

    1. Remond Moningka, et al. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127510.

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