GPR7 antagonist 21a

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Chemical Structure : GPR7 antagonist 21a

Catalog No.: PC-38613Not For Human Use, Lab Use Only.

GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GPR7 antagonist 21a is a highly potent small molecule antagonist of NPBWR1 (GPR7) antagonist with cAMP IC50 of 30 nM, dose-dependently increased [125I]-hNPW23 dissociation rate constants from NPBWR1 in kinetic binding assays.

Physicochemical Properties

M.Wt	397.182
Formula	C17H9Cl2F3N4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(2,6-dichloro-4-(1H-pyrazol-4-yl)phenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazole

References

1. Remond Moningka, et al. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127510.

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