GSK-5959 |CAS:901245-65-6 Probechem Biochemicals

Chemical Structure : GSK-5959

CAS No.: 901245-65-6

GSK-5959 (GSK5959, GSK 5959)

Catalog No.: PC-45508Not For Human Use, Lab Use Only.

GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.

Packing	Price	Stock
10 mg	$128	In stock
25 mg	$218	In stock
50 mg	$378	In stock
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Biological Activity

GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.
GSK-5959 shows about 2 logs selectivity over BRPF2/3 and less potent for BRD4 (pIC50<4.3).

Physicochemical Properties

M.Wt	394.4668
Formula	C22H26N4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: < 7.8 mg/mL
Chemical Name/SMILES	Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy-

References

1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.

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GSK-5959 (GSK5959, GSK 5959)

Biological Activity

Physicochemical Properties

References

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