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Chemical Structure : GSK-5959
CAS No.: 901245-65-6
Catalog No.: PC-45508Not For Human Use, Lab Use Only.
GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $218 | In stock | |
| 50 mg | $378 | In stock | |
| 100 mg | Get quote |
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GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.
GSK-5959 shows about 2 logs selectivity over BRPF2/3 and less potent for BRD4 (pIC50<4.3).
| M.Wt | 394.4668 | |
| Formula | C22H26N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: < 7.8 mg/mL |
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| Chemical Name/SMILES |
Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxy- |
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1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.
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