Chemical Structure : GSK-7975A
CAS No.:
1253186-56-9
GSK-7975A
(GSK-7975;GSK7975)
Catalog No. : PC-70096Not For Human Use, Lab Use Only.
GSK-7975A (GSK7975A) is a selective CRAC channel blocker that inhibits store-operated Ca(2+) entry (SOCE) with IC50 of 3.4 uM.
Packing Price Stock Quantity 25 mg $198 In stock 0 1 2 3 4 5 50 mg $298 In stock 0 1 2 3 4 5 100 mg $488 In stock 0 1 2 3 4 5 200 mg Get quote 0 1 2 3 4 5 1 g Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-7009601
Biological Activity
GSK-7975A (GSK7975A) is a selective CRAC channel blocker that inhibits store-operated Ca(2+) entry (SOCE) with IC50 of 3.4 uM.
Physicochemical Properties
M.Wt
397.305
Formula
C18H12F5N3O2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2,6-difluoro-N-(1-(4-hydroxy-2-(trifluoromethyl)benzyl)-1H-pyrazol-3-yl)benzamide
References
1. Gerasimenko JV, et al. Proc Natl Acad Sci U S A.
2. Rice LV, et al. Eur J Pharmacol.
3. Derler I, et al. Cell Calcium.
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