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GSK040

Chemical Structure : GSK040

CAS No.: 2752331-09-0

GSK040 (GSK-040)

Catalog No.: PC-72181Not For Human Use, Lab Use Only.

GSK040 (GSK-040) is a potent, highly selective BET BD2 inhibitor with pIC50 of 8.3 (BRD4 BD2), 5000-fold selectivity over BD1.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GSK040 (GSK-040) is a potent, highly selective BET BD2 inhibitor with pIC50 of 8.3 (BRD4 BD2), 5000-fold selectivity over BD1.

Physicochemical Properties

M.Wt 502.615
Formula C29H34N4O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Month
Shipping
Solubility

Chemical Name/SMILES

References

1. Rianjongdee F, et al. J Med Chem. 2021 Aug 12;64(15):10806-10833.

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