Chemical Structure : GSK1016790A
CAS No.:
942206-85-1
GSK1016790A
(GSK-1016790A, GSK 1016790A)
Catalog No. : PC-45654Not For Human Use, Lab Use Only.
GSK1016790A is a potent TRPV4 channel agonist, induces Ca2+ influx in HEK cells expressing human TRPV4 with EC50 of 2.1 nM.
Packing Price Stock Quantity 5 mg $78 In stock 0 1 2 3 4 5 10 mg $118 In stock 0 1 2 3 4 5 25 mg $218 In stock 0 1 2 3 4 5 50 mg $348 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4565401
Biological Activity
GSK1016790A is a potent TRPV4 channel agonist, induces Ca2+ influx in HEK cells expressing human TRPV4 with EC50 of 2.1 nM.
Physicochemical Properties
M.Wt
655.613
Formula
C28H32Cl2N4O6S2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 33 mg/mL
Chemical Name/SMILES
Benzo[b]thiophene-2-carboxamide, N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbonyl]-3-methylbutyl]-
References
1. Thorneloe KS, et al. J Pharmacol Exp Ther.
2. Rajasekhar P, et al. J Biol Chem.
3. Hong Z, et al. Mol Neurobiol.
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