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GSK145A

Chemical Structure : GSK145A

CAS No.: 1609945-27-8

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GSK145A (GSK 145A, GSK-145A)

Catalog No.: PC-35105Not For Human Use, Lab Use Only.

GSK145A is a small molecule inhibitor of SUMO-conjugating enzyme E2 with IC50 of 12.5 uM, GSK145A is competitive with the sumoylation of the TRPS1 peptide substrates..

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Purity & Documentation Purity: 98.5% (HPLC) Select Batch:

Biological Activity

GSK145A is a small molecule inhibitor of SUMO-conjugating enzyme E2 with IC50 of 12.5 uM, GSK145A is competitive with the sumoylation of the TRPS1 peptide substrates.

Physicochemical Properties

M.Wt 454.593
Formula C23H30N6O2S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-5-amino-N-(4-methoxyphenyl)-2-((6-methyl-2-((2-(thiophen-2-yl)ethyl)amino)pyrimidin-4-yl)amino)pentanamide

References

1. Brandt M, et al. Assay Drug Dev Technol. 2013 Jun;11(5):308-25.

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