GSK145A | SUMOylation inhibitor | Probechem Biochemicals

Chemical Structure : GSK145A

CAS No.: 1609945-27-8

GSK145A (GSK 145A, GSK-145A)

Catalog No.: PC-35105Not For Human Use, Lab Use Only.

GSK145A is a small molecule inhibitor of SUMO-conjugating enzyme E2 with IC50 of 12.5 uM, GSK145A is competitive with the sumoylation of the TRPS1 peptide substrates..

Packing	Price	Stock
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5 mg	$388	In stock
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Biological Activity

GSK145A is a small molecule inhibitor of SUMO-conjugating enzyme E2 with IC50 of 12.5 uM, GSK145A is competitive with the sumoylation of the TRPS1 peptide substrates.

Physicochemical Properties

M.Wt	454.593
Formula	C23H30N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-5-amino-N-(4-methoxyphenyl)-2-((6-methyl-2-((2-(thiophen-2-yl)ethyl)amino)pyrimidin-4-yl)amino)pentanamide

References

1. Brandt M, et al. Assay Drug Dev Technol. 2013 Jun;11(5):308-25.

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GSK145A (GSK 145A, GSK-145A)

Biological Activity

Physicochemical Properties

References

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