GSK1482160 | P2X7 NAM | Probechem Biochemicals

Chemical Structure : GSK1482160

CAS No.: 1001389-72-5

GSK1482160 (GSK-1482160)

Catalog No.: PC-22645Not For Human Use, Lab Use Only.

GSK1482160 is an orally available allosteric P2X7 receptor negative allosteric modulator (NAM) with pIC50 of 8.5 and 6.5 for human and rat P2X7R respectively.

Packing	Price	Stock
10 mg	$138	In stock
25 mg	$248	In stock
50 mg	$398	In stock
100 mg		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

GSK1482160 is an orally available allosteric P2X7 receptor negative allosteric modulator (NAM) with pIC50 of 8.5 and 6.5 for human and rat P2X7R respectively.

Physicochemical Properties

M.Wt	334.72
Formula	C14H14ClF3N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-{[2-chloro-3-(trifluoromethyl)phenyl]methyl}-1-methyl-5-oxo-L-prolinamide

References

1. Ali Z, et al. Br J Clin Pharmacol. 2013 Jan;75(1):197-207.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com

GSK1482160 (GSK-1482160)

Biological Activity

Physicochemical Properties

References

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

Get Quote

* Indicates a Required FieldYour information is safe with us.