Catalog No.: PC-27046Not For Human Use, Lab Use Only.
GSK1820795A is a potent, specific antagonist of G-protein-coupled receptor GPR132 (G2A), blocks agonist-induced association of hGPR132 with β-arrestin with pIC50 of 7.8, also is a dual angiotensin AT1 antagonist and PPARγ modulator.
GSK1820795A is a potent, specific antagonist of G-protein-coupled receptor GPR132 (G2A), blocks agonist-induced association of hGPR132 with β-arrestin with pIC50 of 7.8, also is a dual angiotensin AT1 antagonist and PPARγ modulator.
GSK1820795A does not antagonize free fatty acid receptor FFA2.
GSK1820795A blocks rGPR132.
GSK1820795A blocks activation of yeast cells expressing hGPR132a by N‐acylamides.
