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Chemical Structure : GSK205 derivative 16-8
Catalog No.: PC-62628Not For Human Use, Lab Use Only.
GSK205 derivative 16-8 is a specific small molecule dual-inhibitor of TRPV4 and TRPA1 with IC50 of 0.45 and 0.41 uM, respectively.
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GSK205 derivative 16-8 is a specific small molecule dual-inhibitor of TRPV4 and TRPA1 with IC50 of 0.45 and 0.41 uM, respectively.
GSK205 derivative 16-8 displays no inhibitory potency toward TRPV1, TRPV2 and TRPV3.
GSK205 derivative 16-8 effectively attenuates formalin-evoked trigeminal irritant pain in model of acute pancreatitis.
| M.Wt | 399.556 | |
| Formula | C25H25N3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Kanju P, et al. Sci Rep. 2016 Jun 1;6:26894.
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