GSK217 | BET BD2 inhibitor | Probechem Biochemicals

Chemical Structure : GSK217

Catalog No.: PC-72184Not For Human Use, Lab Use Only.

GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

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Biological Activity

GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

M.Wt	360.421
Formula	C20H20N6O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((1H-indol-4-yl)methyl)-N-ethyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide

1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281.