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GSK217

Chemical Structure : GSK217

CAS No.: 2748687-92-3

GSK217 (GSK-217)

Catalog No.: PC-72184Not For Human Use, Lab Use Only.

GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

Physicochemical Properties

M.Wt 360.421
Formula C20H20N6O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Month
Shipping
Solubility

Chemical Name/SMILES

References

1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281.

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