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Chemical Structure : GSK2239633A
Catalog No.: PC-73262Not For Human Use, Lab Use Only.
GSK2239633A is a potent, allosteric CC-chemokine receptor 4 (CCR4) antagonist with pIC50 of 7.83 in 35S-GTPγS competition assay.
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GSK2239633A is a potent, allosteric CC-chemokine receptor 4 (CCR4) antagonist with pIC50 of 7.83 in 35S-GTPγS competition assay.
GSK2239633A binds to CCR4 at an intracellular allosteric site denoted site II. GSK2239633A inhibits thymus activation-regulated chemokine (TARC) -induced F-actin polymerization in human whole blood.
| M.Wt | 549.06 | |
| Formula | C24H25ClN4O5S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Procopiou PA, et al. J Med Chem. 2013 Mar 14;56(5):1946-60.
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