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Chemical Structure : GSK2795039
CAS No.: 1415925-18-6
Catalog No.: PC-45569Not For Human Use, Lab Use Only.
GSK2795039 (GSK 2795039) is a potent and selective inhibitor of NOX2 (NADPH oxidase 2) with pIC50 of 6.57.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $188 | In stock | |
| 10 mg | $298 | In stock | |
| 25 mg | $498 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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GSK2795039 (GSK 2795039) is a potent and selective inhibitor of NOX2 (NADPH oxidase 2) with pIC50 of 6.57.
GSK-2795039 exhibits good selectivity for NOX2 over other NOX isoforms, xanthine oxidase and eNOS.
GSK-2795039 abolishes the production of ROS by activated NOX2 enzyme in a paw inflammation model of acute pancreatitis.
| M.Wt | 450.5565 | |
| Formula | C23H26N6O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 32 mg/mL |
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| Chemical Name/SMILES |
1H-Pyrazole-3-sulfonamide, N-[3-(2,3-dihydro-1-methyl-1H-indol-6-yl)-1-(1-methylethyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-methyl- |
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1. Hirano K, et al. Antioxid Redox Signal. 2015 Aug 10;23(5):358-74.
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