GSK3326595 | PRMT5 inhibitor | Probechem Biochemicals

Chemical Structure : GSK3326595

CAS No.: 1616392-22-3

Catalog No.: PC-42405Not For Human Use, Lab Use Only.

Pemrametostat (GSK3326595, EPZ015938) is a potent, selective, reversible and orally active PRMT5 inhibitor with IC50 of 22 nM.

Packing	Price	Stock
10 mg	$68	In stock
25 mg	$118	In stock
50 mg	$198	In stock
100 mg	$328	In stock
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Biological Activity

Pemrametostat (GSK3326595, EPZ015938) is a potent, selective, reversible and orally active PRMT5 inhibitor with IC50 of 22 nM.

M.Wt	452.54928
Formula	C24H32N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	DMSO: ≥ 30 mg/mL
Chemical Name/SMILES	4-Pyrimidinecarboxamide, 6-[(1-acetyl-4-piperidinyl)amino]-N-[(2S)-3-(3,4-dihydro-2(1H)-isoquinolinyl)-2-hydroxypropyl]-

1. Drew Rasco, et al. Abstract CT038, AACR. DOI: 10.1158/1538-7445.

2. Patent WO 2016022605 A1, Formula A.