GSK3527497 | TRPV4 inhibitor | Probechem Biochemicals

Chemical Structure : GSK3527497

GSK3527497 (GSK-3527497)

Catalog No.: PC-73096Not For Human Use, Lab Use Only.

GSK3527497 (GSK-3527497) is a potent, selective TRPV4 inhibitor with IC50 of 12 nM (hTRPV4).

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Biological Activity

GSK3527497 (GSK-3527497) is a potent, selective TRPV4 inhibitor with IC50 of 12 nM (hTRPV4).
GSK3527497 is a pre-clinical candidate for treatment of diseases resulting from TRPV4 activation.

Physicochemical Properties

M.Wt	426.847
Formula	C17H16ClFN4O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-(((3S,4S)-4-(Aminomethyl)-1-((5-chloropyridin-2-yl)-sulfonyl)-4-hydroxypyrrolidin-3-yl)oxy)-2-fluorobenzonitrile

References

1. Carl A Brooks, et al. J Med Chem. 2019 Oct 24;62(20):9270-9280.

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GSK3527497 (GSK-3527497)

Biological Activity

Physicochemical Properties

References

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