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GSK5182

Chemical Structure : GSK5182

CAS No.: 877387-37-6

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GSK5182 (GSK-5182)

Catalog No.: PC-72965Not For Human Use, Lab Use Only.

GSK5182 (GSK-5182) is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with IC50 of 79 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GSK5182 (GSK-5182) is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with IC50 of 79 nM.
GSK5182 displays little to no activities against other nuclear receptors, including ERRα or ERα.

Physicochemical Properties

M.Wt 417.549
Formula C27H31NO3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

100 mM in DMSO (41.7 mg/mL)
Chemical Name/SMILES

(Z)-4-(1-(4-(2-(dimethylamino)ethoxy)phenyl)-5-hydroxy-2-phenylpent-1-en-1-yl)phenol

References

1. Kim DK, et al. J Biol Chem. 2011 Nov 4;286(44):38035-38042.

2. Zhang Y, et al. Biochem J. 2015 Sep 1;470(2):181-93.

3. Xie YB, et al. J Biol Chem. 2009 Oct 16;284(42):28762-74.

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