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Chemical Structure : GSK5182
CAS No.: 877387-37-6
Catalog No.: PC-72965Not For Human Use, Lab Use Only.
GSK5182 (GSK-5182) is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with IC50 of 79 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $198 | In stock | |
| 100 mg | $498 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
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GSK5182 (GSK-5182) is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with IC50 of 79 nM.
GSK5182 displays little to no activities against other nuclear receptors, including ERRα or ERα.
| M.Wt | 417.549 | |
| Formula | C27H31NO3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
100 mM in DMSO (41.7 mg/mL) |
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| Chemical Name/SMILES |
(Z)-4-(1-(4-(2-(dimethylamino)ethoxy)phenyl)-5-hydroxy-2-phenylpent-1-en-1-yl)phenol |
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1. Kim DK, et al. J Biol Chem. 2011 Nov 4;286(44):38035-38042.
2. Zhang Y, et al. Biochem J. 2015 Sep 1;470(2):181-93.
3. Xie YB, et al. J Biol Chem. 2009 Oct 16;284(42):28762-74.
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