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Chemical Structure : GSK549
Catalog No.: PC-72180Not For Human Use, Lab Use Only.
GSK549 (GSK-549) is a potent, highly selective, BD2 domain-selective BET inhibitor with pIC50 of 7.8 (BRD4 BD2), 1150-fold selectivity over BD1.
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GSK549 (GSK-549) is a potent, highly selective, BD2 domain-selective BET inhibitor with pIC50 of 7.8 (BRD4 BD2), 1150-fold selectivity over BD1.
| M.Wt | 366.421 | |
| Formula | C20H22N4O3 | |
| Appearance | Solid | |
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1. Seal JT, et al. J Med Chem. 2020 Sep 10;63(17):9093-9126.
2. Harrison LA, et al. J Med Chem. 2021 Aug 12;64(15):10742-10771.
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