Chemical Structure : GSK591
CAS No.:
1616391-87-7
GSK591
(EPZ015866, GSK-591, GSK3203591)
Catalog No. : PC-42097Not For Human Use, Lab Use Only.
GSK591 (EPZ015866, GSK3203591) is a potent, selective protein methyltransferase 5 (PRMT5) inhibitor with IC50 of 4 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4209701
Biological Activity
GSK591 (EPZ015866, GSK3203591) is a potent, selective protein methyltransferase 5 (PRMT5 ) inhibitor with IC50 of 4 nM.
Physicochemical Properties
M.Wt
380.4833
Formula
C22H28N4O2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
4-Pyridinecarboxamide, 2-(cyclobutylamino)-N-[(2S)-3-(3,4-dihydro-2(1H)-isoquinolinyl)-2-hydroxypropyl]-
References
1. Duncan KW, et al. ACS Med Chem Lett.
2. Gerhart SV, et al. Sci Rep.
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