Chemical Structure : GSK690
Catalog No.: PC-61745Not For Human Use, Lab Use Only.
GSK690 is a reversible, mechanism based inhibitor of lysine specific demethylase 1 (LSD1, KDM1A) with IC50 of 37 nM, binding Kd value of 9 nM.
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GSK690 is a reversible, mechanism based inhibitor of lysine specific demethylase 1 (LSD1, KDM1A) with IC50 of 37 nM, binding Kd value of 9 nM.
M.Wt | 369.468 | |
Formula | C24H23N3O | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Mould DP, et al. J Med Chem. 2017 Sep 11. doi: 10.1021/acs.jmedchem.7b00462.
2. Mould DP, et al. Bioorg Med Chem Lett. 2017 Oct 15;27(20):4755-4759.
3. McGrath JP, et al. Cancer Res. 2016 Apr 1;76(7):1975-88.
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