GSK789 | BET BD1 inhibitor | Probechem Biochemicals

Chemical Structure : GSK789

GSK789 (GSK-789)

Catalog No.: PC-72470Not For Human Use, Lab Use Only.

GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.

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Biological Activity

GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.

Physicochemical Properties

M.Wt	463.582
Formula	C26H33N5O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(3R,4R)-N-cyclohexyl-4-((5-(furan-2-yl)-3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)-1-methylpiperidine-3-carboxamide

References

1. Robert J Watson, et al. J Med Chem. 2020 Sep 10;63(17):9045-9069.

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GSK789 (GSK-789)

Biological Activity

Physicochemical Properties

References

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