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Chemical Structure : GSK789
Catalog No.: PC-72470Not For Human Use, Lab Use Only.
GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.
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GSK789 (GSK-789) is a potent, cell-permeable, and highly selective inhibitor of the first bromodomains (BD1) of the BET family with IC50 of 20 nM BRD4 BD1, 1500-fold selectivity over BD2.
| M.Wt | 463.582 | |
| Formula | C26H33N5O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Robert J Watson, et al. J Med Chem. 2020 Sep 10;63(17):9045-9069.
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