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Chemical Structure : GSK852
Catalog No.: PC-72183Not For Human Use, Lab Use Only.
GSK852 (GSK-852) is a highly potent, second bromodomain (BD2)-selective BET inhibitor with pIC50 7.9 (BRD4 BD2), 1260-fold selectivity over BRD4 BD1.
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GSK852 (GSK-852) is a highly potent, second bromodomain (BD2)-selective BET inhibitor with pIC50 7.9 (BRD4 BD2), 1260-fold selectivity over BRD4 BD1.
GSK852 demonstrates highly soluble with good in vivo rat and dog pharmacokinetics.
| M.Wt | 406.482 | |
| Formula | C24H26N2O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Simon C C Lucas, et al. J Med Chem. 2021 Aug 12;64(15):10711-10741.
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