Chemical Structure : GSK8612
CAS No.:
2361659-62-1
GSK8612
(GSK-8612)
Catalog No. : PC-38171Not For Human Use, Lab Use Only.
GSK8612 (GSK-8612) is a highly selective, potent TBK1 inhibitor, inhibits recombinant TBK1 with pIC50 of 6.8 in biochemical functional assays.
Packing Price Stock Quantity 5 mg $88 In stock 0 1 2 3 4 5 10 mg $128 In stock 0 1 2 3 4 5 25 mg $218 In stock 0 1 2 3 4 5 50 mg $368 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-3817101
Biological Activity
GSK8612 (GSK-8612) is a highly selective, potent TBK1 inhibitor, inhibits recombinant TBK1 with pIC50 of 6.8 in biochemical functional assays.
Physicochemical Properties
M.Wt
520.329
Formula
C17H17BrF3N7O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
4-((5-bromo-2-((3-methyl-1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl)amino)pyrimidin-4-ylamino)methyl)benzenesulfonamide
References
1. Thomson DW, et al. ACS Med Chem Lett.
2. Chen S, et al. Am J Transl Res.
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