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GSK902056A

Chemical Structure : GSK902056A

CAS No.: 913642-05-4

GSK902056A (GSK-902056A)

Catalog No.: PC-26112Not For Human Use, Lab Use Only.

GSK902056A is a highly potent inhibitor of serine/threonine kinase PKN3 with Kdapp of 1 nM, potently engaged PKN3 in cells with IC50 of 79 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GSK902056A is a highly potent inhibitor of serine/threonine kinase PKN3 with Kdapp of 1 nM, potently engaged PKN3 in cells with IC50 of 79 nM.

Physicochemical Properties

M.Wt 371.40
Formula C17H21N7O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoethoxy)-1-ethyl-1H-imidazo[4,5-c]pyridin-4-yl)-2-methylbut-3-yn-2-ol

References

1. Maria Reinecke, et al. Nat Chem Biol. 2024 May;20(5):577-585.

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