GlpG inhibitor 11 | Probechem Biochemicals

Chemical Structure : GlpG inhibitor 11

GlpG inhibitor 11 (Rhomboid protease inhibitor)

Catalog No.: PC-60493Not For Human Use, Lab Use Only.

A potent, selective, reversible rhomboid proteases inhibitor with Ki of 45 nM for GlpG .

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Biological Activity

A potent, selective, reversible rhomboid proteases inhibitor with Ki of 45 nM for GlpG ; does not inhibit most of the human serine hydrolases with the exception of PRCP and DPP7; potently inhibits endogenous GlpG in living E.coli. with IC50 of 2.7 nM.

Physicochemical Properties

M.Wt	855.015
Formula	C39H62N14O8
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-(2-((S)-1-(((S)-3,4-dioxo-4-((4-phenylbutoxy)amino)butan-2-yl)amino)-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl)hydrazinyl)-5-guanidino-N-((S)-1-(((S)-1-guanidino-5,6-dioxoheptan-4-yl)amino)-3-methyl-1-oxobutan-2-yl)pentanamide

References

1. Tichá A, et al. Cell Chem Biol. 2017 Dec 21;24(12):1523-1536.e4.

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GlpG inhibitor 11 (Rhomboid protease inhibitor)

Biological Activity

Physicochemical Properties

References

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