Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-Nuclear Receptor/Transcription Factor-HIF/HIF Prolyl-hydroxylase-HIF2α-IN-1
HIF2α-IN-1

Chemical Structure : HIF2α-IN-1

CAS No.: 1799948-06-3

HIF2α-IN-1

Catalog No.: PC-45759Not For Human Use, Lab Use Only.

A potent HIF-2α inhibitor with IC50 of <500 nM in HIF-2α scintillation proximity assay. .

Packing Price Stock Quantity
10 mg $800 In stock
25 mg $1680 In stock

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent HIF-2α inhibitor with IC50 of <500 nM in HIF-2α scintillation proximity assay.

Physicochemical Properties

M.Wt 405.2961
Formula C16H8F5NO4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

Benzonitrile, 3-[[(3R)-4-(difluoromethyl)-2,2-difluoro-2,3-dihydro-3-hydroxy-1,1-dioxidobenzo[b]thien-5-yl]oxy]-5-fluoro-

References

1. Bruick Richard Keith, et al. From PCT Int. Appl. (2016), WO 2016057242 A1 20160414.

2. Dixon Darryl David, et al. From PCT Int. Appl. (2015), WO 2015095048 A1 20150625.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: