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HKMTI-1-248

Chemical Structure : HKMTI-1-248

CAS No.: 1910102-10-1

HKMTI-1-248

Catalog No.: PC-23904Not For Human Use, Lab Use Only.

HKMTI-1-248 is a potent and selective G9a/GLP inhibitor with IC50 of 13 nM (G9a), equipotent against G9a and GLP (G9a-like protein, EHMT1).

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

HKMTI-1-248 is a potent and selective G9a/GLP inhibitor with IC50 of 13 nM (G9a), equipotent against G9a and GLP (G9a-like protein, EHMT1).

Physicochemical Properties

M.Wt 489.66
Formula C29H39N5O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(1-benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinolin-4-amine

References

1. Srimongkolpithak N, et al. Medchemcomm. 2014 Dec 19;5(12):1821-1828.

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