HTL0041178 | GPR52 agonist | Probechem Biochemicals

Chemical Structure : HTL0041178

HTL0041178 (HTL 0041178)

Catalog No.: PC-20325Not For Human Use, Lab Use Only.

HTL0041178 is a potent GPR52 agonist with EC50 of 27.5 nM (human or rat GPR52).

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Biological Activity

HTL0041178 is a potent GPR52 agonist with EC50 of 27.5 nM (human or rat GPR52).
HTL0041178 exhibits a promising pharmacokinetic (PK) profile, and oral activity in rodent preclinical models.
HTL0041178 (10 mg/kg, p.o.) caused a dose-related reduction in d-amphetamine-stimulated hyperlocomotion in rats.

Physicochemical Properties

M.Wt	390.34
Formula	C19H14F4N4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(2-(3-fluoro-5-(trifluoromethyl)benzyl)pyridin-4-yl)-1,5,6,7-tetrahydro-4H-pyrazolo[4,3-c]pyridin-4-one

References

1. Patent WO2021090030

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HTL0041178 (HTL 0041178)

Biological Activity

Physicochemical Properties

References

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