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I-BET282E

Chemical Structure : I-BET282E

CAS No.: 2885162-99-0

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I-BET282E (I-BET282 mesylate)

Catalog No.: PC-20161Not For Human Use, Lab Use Only.

I-BET282E (I-BET282 mesylate) is the mesylate salt of I-BET282, I-BET282 is a potent and selective pan-inhibitor of bromodomain and extra terminal (BET) proteins.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    I-BET282E (I-BET282 mesylate) is the mesylate salt of I-BET282 (Cat# PC-20162), I-BET282 is a potent and selective pan-inhibitor of bromodomain and extra terminal (BET) proteins.
    I-BET282E (I-BET282 mesylate) (3 mg/kg, p.o.) shows in vivo efficacy in the rat collagen-induced arthritis (CIA) model.

    Physicochemical Properties

    M.Wt 546.64
    Formula C26H34N4O7S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R)-4-(8-methoxy-1-(1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole methanesulfonate

    References

    1. Katherine L Jones, et al. J Med Chem. 2021 Aug 26;64(16):12200-12227.

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