IDOR-1136-517

Chemical Structure : IDOR-1136-517

Catalog No.: PC-24077Not For Human Use, Lab Use Only.

IDOR-1136-5177 is a highly potent, selective CCR8 antagonist with IC50 of 2 nM (hCCR8).

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Biological Activity

IDOR-1136-5177 is a highly potent, selective CCR8 antagonist with IC50 of 2 nM (hCCR8).
IDOR-1136-5177 potently inhibits the CCR8 receptor of the macaque and the dog (IC50=5/4 nM) but is inactive against mouse and rat CCR8.

Physicochemical Properties

M.Wt	390.51
Formula	C18H26N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(cis-3-(2-amino-6-(isopropylamino)pyrimidin-4-yl)cyclobutyl)-5,6-dimethylpyridine-3 sulfonamide

References

1. Diethelm S, et al. ChemMedChem. 2025 Feb 23:e202400968.

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IDOR-1136-517

Biological Activity

Physicochemical Properties

References

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