ISAM-MM101 | CB1R antagonist | Probechem Biochemicals

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Chemical Structure : ISAM-MM101

ISAM-MM101 (CB1R antagonist 24a)

Catalog No.: PC-28685Not For Human Use, Lab Use Only.

ISAM-MM101 (CB1R antagonist 24a) is a potent, selective and peripherally directed CB1 receptor (CB1R) antagonist with Ki of 115 nM, shows high CB1R/CB2R selectivity.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

ISAM-MM101 (CB1R antagonist 24a) is a potent, selective and peripherally directed CB1 receptor (CB1R) antagonist with Ki of 115 nM, shows high CB1R/CB2R selectivity.
ISAM-MM101 exhibits robust functional activity in a biologically relevant model of metabolic dysfunction.
ISAM-MM101 restores insulin-stimulated Akt phosphorylation and significantly enhances lipolytic activity in insulin-resistant, lipid-hypertrophied adipocytes.

Physicochemical Properties

M.Wt	704.86
Formula	C28H33Cl3IN5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(2-(tert-butylamino)-2-oxoethyl)-4-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl)-1-methylpiperazin-1-ium iodide

References

1. Azuaje J, et al. ACS Omega. 2026 Oct 13;11(42):65239-65258.

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ISAM-MM101 (CB1R antagonist 24a)

Biological Activity

Physicochemical Properties

References

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