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JKC-363

Chemical Structure : JKC-363

CAS No.: 436083-30-6

JKC-363 (JKC363)

Catalog No.: PC-22664Not For Human Use, Lab Use Only.

JKC-363 (JKC363) is a highly potent, selective melanocortin MC4 receptor antagonist with IC50 of 0.5 nM, 90-fold selective over MC3 receptor.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

JKC-363 (JKC363) is a highly potent, selective melanocortin MC4 receptor antagonist with IC50 of 0.5 nM, 90-fold selective over MC3 receptor.

Physicochemical Properties

M.Wt 1506.71
Formula C69H91N19O16S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(cyclic [Mpr11, D-Nal14, Cys18, Asp22-NH2]-beta-MSH11-22

References

1. Kim RY, et al. Biochem Biophys Res Commun. 2005 Apr 22;329(4):1178-85.

2. Doghman M, et al. Endocrinology. 2004 Feb;145(2):541-7.

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