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Chemical Structure : Jaspamycin
Catalog No.: PC-23310Not For Human Use, Lab Use Only.
Jaspamycin (7-CN-7-C-Ino) is a potent activator of Trypanosoma brucei PKA (TbPKA), binding to the R site (PKAR) with EC50 of 6.5 nM and Kd of 8 nM in Trypanosoma brucei, also inhibits hepatocellular carcinoma progression via trageting metastasis-associated protein 3 (MTA3).
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Jaspamycin (7-CN-7-C-Ino) is a potent activator of Trypanosoma brucei PKA (TbPKA), binding to the R site (PKAR) with EC50 of 6.5 nM and Kd of 8 nM in Trypanosoma brucei, also inhibits hepatocellular carcinoma progression via trageting metastasis-associated protein 3 (MTA3).
| M.Wt | 292.25 | |
| Formula | C12H12N4O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Sabine Bachmaier, et al. Nat Commun. 2019 Mar 29;10(1):1421.
2. Liu Y, et al. Sci Rep. 2024 Oct 25;14(1):25294.
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