KDM5A covalent inhibitor N71 | Probechem Biochemicals

Chemical Structure : KDM5A covalent inhibitor N71

KDM5A covalent inhibitor N71 (KDM5A inhibitor N71)

Catalog No.: PC-35800Not For Human Use, Lab Use Only.

KDM5A covalent inhibitor N71 is an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481, >20-fold selectivity over KDM4A..

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Biological Activity

KDM5A covalent inhibitor N71 is an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481, >20-fold selectivity over KDM4A.

Physicochemical Properties

M.Wt	522.664
Formula	C28H34N4O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-2-((3-(4-(dimethylamino)but-2-enamido)phenyl)(2-(piperidin-1-yl)ethoxy)methyl)thieno[3,2-b]pyridine-7-carboxylic acid

References

1. Horton JR, et al. J Med Chem. 2018 Nov 15. doi: 10.1021/acs.jmedchem.8b01219.

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KDM5A covalent inhibitor N71 (KDM5A inhibitor N71)

Biological Activity

Physicochemical Properties

References

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