KHK-IN-8 |CAS:1303469-70-6 Probechem Biochemicals

Chemical Structure : KHK-IN-8

CAS No.: 1303469-70-6

KHK-IN-8 (Ketohexokinase inhibitor 8)

Catalog No.: PC-43252Not For Human Use, Lab Use Only.

KHK-IN-8 is a potent ketohexokinase (KHK) inhibitor with IC50 of 12 nM, interacts with Asp-27B in the ATP-binding region of KHK, also shows potent cellular KHK inhibition with IC50 of <500 nM.

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Biological Activity

KHK-IN-8 is a potent ketohexokinase (KHK) inhibitor with IC50 of 12 nM, interacts with Asp-27B in the ATP-binding region of KHK, also shows potent cellular KHK inhibition with IC50 of <500 nM.

Physicochemical Properties

M.Wt	422.5497
Formula	C21H26N8S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Pyrimido[5,4-d]pyrimidine-4,8-diamine, N8-(cyclopropylmethyl)-N4-[2-(methylthio)phenyl]-2-(1-piperazinyl)-

References

1. Maryanoff BE, et al. ACS Med Chem Lett. 2011 Apr 18;2(7):538-43.

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KHK-IN-8 (Ketohexokinase inhibitor 8)

Biological Activity

Physicochemical Properties

References

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