Gintemetostat (KTX-1001) | NSD2 inhibitor

Chemical Structure : KTX-1001

CAS No.: 2604513-16-6

Catalog No.: PC-21038Not For Human Use, Lab Use Only.

Gintemetostat (KTX-1001) is a potent, selective histone methyltransferase NSD2 (WHSC1, MMSET) inhibitor targeting the catalytic SET domain.

Packing	Price	Stock
2 mg	$158	In stock
5 mg	$258	In stock
10 mg	$398	In stock
25 mg	$598	In stock
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100 mg		Get quote

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Biological Activity

Gintemetostat (KTX-1001) is a potent, selective histone methyltransferase NSD2 (WHSC1, MMSET) inhibitor targeting the catalytic SET domain.

M.Wt	546.53
Formula	C25H26F4N8O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-1-((R)-3-amino-1-(4-((6-amino-9H-purin-9-yl)methyl)-6-(2,5-difluoro-4-methoxyphenyl)pyridin-3-yl)piperidin-3-yl)-2,2-difluoroethan-1-ol

1. Patent WO2021026803 A1