KUNG94 | Grp94 inhibitor | Probechem Biochemicals

Chemical Structure : KUNG94

KUNG94 (KUNG-94, KUNG 94)

Catalog No.: PC-60156Not For Human Use, Lab Use Only.

KUNG94 is a potent, selective Grp94 inhibitor with IC50 of 8 nM.

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Biological Activity

KUNG94 is a potent, selective Grp94 inhibitor with IC50 of 8 nM.
KUNG94 displays 10-fold selecticity over Hsp90α.
KUNG94 shows antiproliferative activity against RPMI8226 cells with Gi50 of 1.4 uM, reduces LRP6 levels and induces apoptosis.

Physicochemical Properties

M.Wt	363.388
Formula	C22H18FNO3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(5-(4-fluorobenzyl)-2,4-dihydroxyphenyl)(isoindolin-2-yl)methanone

References

1. Khandelwal A, et al. ACS Med Chem Lett. 2017 Sep 1;8(10):1013-1018.

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KUNG94 (KUNG-94, KUNG 94)

Biological Activity

Physicochemical Properties

References

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