Keap1-Nrf2 inhibitor 57

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Chemical Structure : Keap1-Nrf2 inhibitor 57

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Catalog No.: PC-23226Not For Human Use, Lab Use Only.

Keap1-Nrf2 inhibitor 57 is a higly potent, noncovalent Keap1-Nrf2 inhibitor with Ki of 13 nM in FP assays, binds the Keap1 Kelch domain with excellent selectivity over close homologues from the Kelch-like protein family.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Physicochemical Properties

M.Wt	596.63
Formula	C32H25FN4O5S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(2-((3-Cyano-4-fluorophenyl)sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl)-2-(9-methyl-9H-carbazole-4-carboxamido)acetic Acid

References

1. Qin Y, et al. J Med Chem. 2024 Oct 17. doi: 10.1021/acs.jmedchem.4c01221.

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