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LB-102

Chemical Structure : LB-102

CAS No.: 2227154-23-4

LB-102 (LB102)

Catalog No.: PC-23209Not For Human Use, Lab Use Only.

LB-102 is an N-methylated analogue of amisulpride, selective dopamine D(2/3)/5-HT(7) inhibitor, binds to the D2 receptor and 5-HT7 receptor with Ki of 0.85 nM and 31 nM respectively, shows potential for treatment of schizophrenia and other psychiatric disorders.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

LB-102 is an N-methylated analogue of amisulpride, selective dopamine D(2/3)/5-HT(7) inhibitor, binds to the D2 receptor and 5-HT7 receptor with Ki of 0.85 nM and 31 nM respectively, shows potential for treatment of schizophrenia and other psychiatric disorders.

Physicochemical Properties

M.Wt 383.51
Formula C18H29N3O4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-((1-ethylpyrrolidin-2-yl)methyl)-5-(ethylsulfonyl)-2-methoxy-4-(methylamino)benzamide

References

1. Biernat L, et al. Psychopharmacology (Berl). 2022 Sep;239(9):3009-3018.

2. Grattan V, et al. ACS Omega. 2019 Aug 15;4(9):14151-14154.

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