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Chemical Structure : LEI-102
Catalog No.: PC-20746Not For Human Use, Lab Use Only.
LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.
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LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.
LEI-102 is more potent than the selective CB2R agonists APD371 and HU308.
LEI-102 activates CB2R as a partial agonist (Emax 76 ± 1%) with a pEC50 value of 6.9 in G protein activation assays.
| M.Wt | 454.55 | |
| Formula | C25H31FN4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Xiaoting Li, et al. Nat Commun. 2023 Mar 15;14(1):1447.
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