LEI-102 | CB2R agonist | Probechem Biochemicals

Chemical Structure : LEI-102

LEI-102 (LEI 102)

Catalog No.: PC-20746Not For Human Use, Lab Use Only.

LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.

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Biological Activity

LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.
LEI-102 is more potent than the selective CB2R agonists APD371 and HU308.
LEI-102 activates CB2R as a partial agonist (Emax 76 ± 1%) with a pEC50 value of 6.9 in G protein activation assays.

Physicochemical Properties

M.Wt	454.55
Formula	C25H31FN4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C1N(CC(C)C)C(CN1CC2=CC=C(C3=NC(CNC4CCOCC4)=C(F)C=C3)C=C2)=O

References

1. Xiaoting Li, et al. Nat Commun. 2023 Mar 15;14(1):1447.

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LEI-102 (LEI 102)

Biological Activity

Physicochemical Properties

References

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