LH168 | WDR5 inhibitor | Probechem Biochemicals

Chemical Structure : LH168

LH168 (LH-168)

Catalog No.: PC-25506Not For Human Use, Lab Use Only.

LH168 is a potent, exquisitely selective WDR5 chemical probe inhibitor with EC50 of 10 nM in cellulo target engagement NanoBRET assays, SPR KD of 1.9 nM.

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Biological Activity

LH168 is a potent, exquisitely selective WDR5 chemical probe inhibitor with EC50 of 10 nM in cellulo target engagement NanoBRET assays, SPR KD of 1.9 nM.

Physicochemical Properties

M.Wt	584.66
Formula	C29H31F3N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-3-((1H-imidazol-1-yl)methyl)-N-(1-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-1-oxopentan-2-yl)-5-(1-ethyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)benzamide

References

1. Lasse Hoffmann, et al. RSC Chem Biol. 2025 Jul 17. doi: 10.1039/d5cb00109a.

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LH168 (LH-168)

Biological Activity

Physicochemical Properties

References

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