LSD1-IN-11p |CAS:2101951-67-9 Probechem Biochemicals

Chemical Structure : LSD1-IN-11p

LSD1-IN-11p

Catalog No.: PC-62840Not For Human Use, Lab Use Only.

LSD1-IN-11p is a potent, reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.

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Biological Activity

LSD1-IN-11p is a potent, reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.
LSD1-IN-11p upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM).
LSD1-IN-11p has moderate oral bioavailability in mice (F%=38%).

Physicochemical Properties

M.Wt	420.473
Formula	C22H24N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-4-(3-(3-aminopiperidine-1-carbonyl)-5-((3-ethylisoxazol-5-yl)methoxy)-1H-pyrazol-1-yl)benzonitrile

References

1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195.

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LSD1-IN-11p

Biological Activity

Physicochemical Properties

References

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