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Chemical Structure : LX-039
Catalog No.: PC-38780Not For Human Use, Lab Use Only.
LX-039 is a novel potent, oral and selective estrogen receptor degrader (SERD) with binding IC50 of 0.99 nM, MCF7 antiproliferation IC50 of 3.76 nM.
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LX-039 is a novel potent, oral and selective estrogen receptor degrader (SERD) with binding IC50 of 0.99 nM, MCF7 antiproliferation IC50 of 3.76 nM.
LX-039 exhibits profound anti-tumor activity, desirable ER antagonistic characteristics combined with favorable pharmacokinetic and preliminary safety properties.
| M.Wt | 480.360 | |
| Formula | C27H20Cl2FNO2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Jianyu Lu, et al. Bioorg Med Chem Lett. 2022 Jun 15;66:128734.
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