Legumain inhibitor 10t

Chemical Structure : Legumain inhibitor 10t

Catalog No.: PC-20813Not For Human Use, Lab Use Only.

Legumain inhibitor 10t is a potent, selective and cellularly active Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 71 nM.

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Biological Activity

Legumain inhibitor 10t is a potent, selective and cellularly active Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 71 nM.
Legumain inhibitor 10t blocks colony formation in both metastatic breast (MCF7) and prostate (PC3) cancer cell lines with IC50 of 5 and 2.5 uM, respectively.

Physicochemical Properties

M.Wt	482.60
Formula	C25H30N4O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C([C@H]1N(S(=O)(C2=CC=C(C3=CC=C(C(C)(C)C)C=C3)C=C2)=O)CCC1)N[C@H](C#N)CC(N)=O

References

1. Kerry A Ness, et al. Bioorg Med Chem Lett. 2015 Dec 1;25(23):5642-5.

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