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Chemical Structure : Lenabasum
Catalog No.: PC-61381Not For Human Use, Lab Use Only.
Lenabasum (Ajulemic acid, IP-751, Anabasum) is a synthetic nonpsychoactive cannabinoid acid with potent analgesic and anti-inflammatory activity in vivo, binds directly and selectively to PPARγ.
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Lenabasum (Ajulemic acid, IP-751, Anabasum) is a synthetic nonpsychoactive cannabinoid acid with potent analgesic and anti-inflammatory activity in vivo, binds directly and selectively to PPARγ.
Lenabasum produces significant antitumor activity and effects its actions primarily via CB(2) receptors.
Lenabasum inhibits interleukin-8 promoter activity in a PPARgamma-dependent manner; significantly suppresses CYP-induced urinary frequency in rats at 10 mg/kg.
| M.Wt | 400.559 | |
| Formula | C25H36O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Recht LD, et al. Biochem Pharmacol. 2001 Sep 15;62(6):755-63.
2. Ambrosio AL, et al. J Biol Chem. 2007 Jun 22;282(25):18625-33.
3. Johnson DR, et al. J Cell Biochem. 2007 Jan 1;100(1):184-90.
4. Hiragata S, et al. Urology. 2007 Jul;70(1):202-8.
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