Chemical Structure : Linagliptin
CAS No.:
668270-12-0
Linagliptin
(BI 1356;BI-1356;BI1356)
Catalog No. : PC-42508Not For Human Use, Lab Use Only.
Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM.
Packing Price Stock Quantity 25 mg $88 In stock 0 1 2 3 4 5 100 mg $158 In stock 0 1 2 3 4 5 200 mg $248 In stock 0 1 2 3 4 5 1 g Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4250801
Biological Activity
Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM.
Physicochemical Properties
M.Wt
472.5422
Formula
C25H28N8O2
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
1H-Purine-2,6-dione, 8-[(3R)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-
References
1. Eckhardt M, et al. J Med Chem.
2. Thomas L, et al. J Pharmacol Exp Ther.
3. Thomas L, et al. J Pharmacol Exp Ther.
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